Efficient, divergent synthesis of cryptophycin unit A analogues.

نویسندگان

  • Kyle L Bolduc
  • Scott D Larsen
  • David H Sherman
چکیده

A flexible and divergent synthesis of cryptophycin unit A analogues is described. This method relies on iridium-catalysed stereo- and enantioselective crotylation and chemoselective one-pot oxidative olefination to access common intermediate . Heck, cross metathesis, and Suzuki-Miyaura reactions are illustrated for the generation of methyl ester unit A analogues .

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عنوان ژورنال:
  • Chemical communications

دوره   شماره 

صفحات  -

تاریخ انتشار 2012